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Georgy I. Kovalev

affiliation not provided to SSRN

SCHOLARLY PAPERS

1

DOWNLOADS

24

TOTAL CITATIONS

0

Scholarly Papers (1)

1.

Discovery of 17-imidazo[1,2-a]pyridinyl-3α-hydroxy-5α-androstanes (17IPAs) as novel potent positive allosteric modulators of the GABAA receptor: Synthesis, in vitro and in silico studies

Number of pages: 21 Posted: 28 Apr 2026
affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Russian Academy of Sciences (RAS), affiliation not provided to SSRN and affiliation not provided to SSRN
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Abstract:

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Neuroactive steroids, allopregnanolone, imidazo[1, 2-a]pyridine, heterosteroids, GABA type A receptors