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Hong-Min Liu

Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies

SCHOLARLY PAPERS

7

DOWNLOADS

315

TOTAL CITATIONS

0

Scholarly Papers (7)

1.

Neddylation‐Dependent LSD1 Destabilization Inhibits the Stemness and Chemoresistance of Gastric Cancer

Number of pages: 40 Posted: 06 Mar 2023
Zhengzhou University - Henan Key Laboratory of Precision Clinical Pharmacy, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, University of California, Irvine - Department of Urology, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, The University of Hong Kong - School of Chinese Medicine, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University - Department of Pharmacy and Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies
Downloads 70 (875,328)

Abstract:

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LSD1, neddylation, UBE2M, stemness, gastric cancer

2.

Design, Synthesis and Biological Evaluation of Novel Indole-Capped Histone Deacetylase 6 Inhibitors as Anti-Gastric Cancer Agents

Number of pages: 45 Posted: 27 Apr 2025
Zhengzhou University, Henan University of Technology, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Henan University of Technology, Henan University of Technology, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies and Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies
Downloads 58 (1,000,027)

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Gastric cancer, HDAC6 inhibitors, Indole-capped, lead optimization

3.

Proapoptotic Effect of WS-299 Induced by NOXA Accumulation and NRF2-Counterbalanced Oxidative Stress Damage Through Targeting RBX1-UBE2M Interaction in Gastric Cancer

Number of pages: 29 Posted: 15 Jan 2022
Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University and Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies
Downloads 57 (989,921)

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RBX1-UBE2M interaction, Nrf2, NOXA, Apoptosis, ROS

4.

Design, Synthesis and Biological Evaluation of Novel Histone Deacetylase 6 Inhibitors Containing Indole-Based Cap Groups

Number of pages: 18 Posted: 29 Jul 2025
Zhengzhou University, Henan University of Technology, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Henan University of Technology, Henan University of Technology, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies and Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies
Downloads 56 (1,010,164)

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HDAC6 inhibitors, indole, lead optimization, gastric cancer

5.

6-Heterocyclic Carboxylic Ester Derivatives of Gliotoxin Lead to LSD1 Inhibitors in Gastric Cancer Cells

Number of pages: 30 Posted: 14 Aug 2022
Zhengzhou University - School of Pharmaceutical Sciences, Zhengzhou University - School of Pharmaceutical Sciences, Zhengzhou University - School of Pharmaceutical Sciences, Zhengzhou University - School of Pharmaceutical Sciences, Zhengzhou University - School of Pharmaceutical Sciences, Zhengzhou University - School of Pharmaceutical Sciences, Zhengzhou University - School of Pharmaceutical Sciences, Zhengzhou University - School of Pharmaceutical Sciences, Zhengzhou University - School of Pharmaceutical Sciences and Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies
Downloads 36 (1,236,159)

Abstract:

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Gliotoxin derivatives, LSD1 inhibitor, Gratric cancer, Antiproliferation, Mobility

6.

Targeting LSD1 Inhibits Gastric Cancer by Reprogramming Macrophages and Restoring T-Cell Response

Number of pages: 30 Posted: 09 Jun 2026
Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University, Zhengzhou University, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, University of Auckland, University of Auckland, The University of Hong Kong - School of Chinese Medicine, Zhengzhou University, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University and Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies
Downloads 24

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Gastric cancer, LSD1, Quinoline-based LSD1 inhibitor, Macrophage polarization, CD8+ T-cell exhaustion

7.

Targeting LSD1 inhibits gastric cancer by reprogramming macrophages and restoring T-cell response

Number of pages: 32 Posted: 15 May 2026
Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University, Zhengzhou University, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, University of Auckland, University of Auckland, The University of Hong Kong - School of Chinese Medicine, Zhengzhou University, Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies, Zhengzhou University and Zhengzhou University - Key Laboratory of Advanced Drug Preparation Technologies
Downloads 14 (1,534,404)

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gastric cancer, LSD1, Quinoline-based LSD1 inhibitor, Macrophage polarization, CD8+ T-cell exhaustion.