Yanan Yu

East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development

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Scholarly Papers (1)

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Function-Oriented Synthesis of Imidazo[1,2-a]Pyrazine and Imidazo[1,2-b]Pyridazine Derivatives as Potent PI3K/mTOR Dual Inhibitors

Posted: 08 Nov 2022
East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, Shanghai University of Engineering Science, East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, Chinese Academy of Sciences (CAS) - State Key Laboratory of Drug Research, East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development and East China Normal University (ECNU) - Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development

Abstract:

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PI3K/mTOR dual inhibitors, Cancer, Antitumor activity, Hepatotoxicity.