default author photo

Hua Yang

Zhengzhou University

100 Science Avenue

Zhengzhou, CO 450001

China

SCHOLARLY PAPERS

3

DOWNLOADS

139

TOTAL CITATIONS

0

Scholarly Papers (3)

1.

Design, Synthesis, and Biological Activity Evaluation of Novel Tubulin Polymerization Inhibitors Based on Pyrimidine Ring Skeletons

Number of pages: 9 Posted: 29 Nov 2022
Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University and Zhengzhou University
Downloads 52 (1,041,696)

Abstract:

Loading...

tubulin, colchicine site, pyrimidine, tubulin inhibitors, antitumor

2.

Design and Synthesis of Cereblon-Based Protac as Novel Potent Degraders of Α/Β-Tubulin

Number of pages: 28 Posted: 30 Aug 2025
Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University and Zhengzhou University
Downloads 45 (1,121,190)

Abstract:

Loading...

tubulin, PROTAC, degrade, drug resistance, CRBN

3.

Design, Synthesis and in Vitro Antitumor Activity Evaluation of a Novel Neddylation Inhibitor

Number of pages: 16 Posted: 22 Nov 2023
Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University, Zhengzhou University and Zhengzhou University
Downloads 42 (1,157,785)

Abstract:

Loading...

Protein degradation, anti-tumor, Neddylation, NAE, NEDD8