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Anna Krupa

Jagiellonian University in Krakow

SCHOLARLY PAPERS

3

DOWNLOADS

145

TOTAL CITATIONS

0

Scholarly Papers (3)

1.

Discovery and Profiling of Novel Multi-Mechanistic Phenylglycinamide Derivatives as Potent Antiseizure and Antinociceptive Drug Candidates

Number of pages: 83 Posted: 17 May 2024
Jagiellonian University Medical College, Jagiellonian University Medical College, affiliation not provided to SSRN, Maria Curie-Sklodowska University, University of Utah, Jagiellonian University in Krakow - Faculty of Pharmacy, Jagiellonian University Medical College, Jagiellonian University Medical College, affiliation not provided to SSRN, University of Utah, University of Utah, Jagiellonian University Medical College, Jagiellonian University Medical College, Medical University of Warsaw, Jagiellonian University in Krakow, Jagiellonian University Medical College, Maria Curie-Sklodowska University, Jagiellonian University Medical College, University of Utah, affiliation not provided to SSRN, Jagiellonian University Medical College and Jagiellonian University Medical College
Downloads 58 (1,000,027)

Abstract:

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hybrid molecules, multi-mechanistic compounds, antiseizure activity, antinociceptive activity, in vitro functional studies, in vitro ADME-Tox studies

2.

High Energy Ball Milling vs. Nano Spray Drying in the Development of Supersaturated Systems Loaded with Bosentan

Number of pages: 35 Posted: 07 Mar 2023
Jagiellonian University in Krakow, University of Lille, Jagiellonian University in Krakow, Jagiellonian University in Krakow, Jagiellonian University in Krakow, Jagiellonian University in Krakow and University of Lille
Downloads 53 (1,031,043)

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bosentan, supersaturation, enabling formulations, solvent evaporation, mechanical activation, poorly soluble drugs

3.

Molecular Phenomena Related to Moisture Uptake in Amorphous Solid Dispersions Loaded with Bosentan Monohydrate and Copovidone

Number of pages: 49 Posted: 08 Jun 2023
affiliation not provided to SSRN, Jagiellonian University in Krakow, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Jagiellonian University in Krakow and affiliation not provided to SSRN
Downloads 34 (1,263,436)

Abstract:

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bosentan hydrate, Kollidon VA64, amorphous drugs, Hydration kinetics, surface wetting, intrinsic dissolution, water sorption, spin-spin relaxation time