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Weige Zhang

Shenyang Pharmaceutical University

Shenyang

China

SCHOLARLY PAPERS

2

DOWNLOADS

59

TOTAL CITATIONS

0

Scholarly Papers (2)

1.

Design, Synthesis and Biological Evaluation of Novel Tubulin-Targeting Agents with a Dual-Mechanism for Polymerization Inhibition and Protein Degradation

Number of pages: 52 Posted: 13 Mar 2024
Shenyang Pharmaceutical University, Shenyang Pharmaceutical University, Shenyang Pharmaceutical University, Shenyang Pharmaceutical University, Shenyang Pharmaceutical University, Shenyang Pharmaceutical University, Chinese Medical University, Chinese Medical University, Shenyang Pharmaceutical University and Shenyang Pharmaceutical University
Downloads 39 (1,222,651)

Abstract:

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Dual-mechanism tubulin-targeting agents, Hydrophobic tagging, Tubulin polymerization inhibition, Protein degradation

2.

Pocket-Based Lead Optimization Strategy for the Design and Synthesis of Tubulin Polymerization Inhibitors

Number of pages: 25 Posted: 16 May 2024
affiliation not provided to SSRN, Shenyang Pharmaceutical University, affiliation not provided to SSRN, Shenyang Pharmaceutical University, affiliation not provided to SSRN, Shenyang Pharmaceutical University, Shenyang Pharmaceutical University and Shenyang Pharmaceutical University
Downloads 20 (1,459,862)

Abstract:

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Microtubule, Colchicine binding site, tubulin polymerization inhibitor