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Gerard J. P. van Westen

Leiden University - Leiden Academic Centre for Drug Research

SCHOLARLY PAPERS

2

DOWNLOADS

162

TOTAL CITATIONS

0

Scholarly Papers (2)

1.

Impact of Cancer-Associated Mutations in CC Chemokine Receptor 2 on Receptor Function and Antagonism

Number of pages: 33 Posted: 03 Nov 2022
Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research and Leiden University - Leiden Academic Centre for Drug Research
Downloads 105 (669,616)

Abstract:

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CC chemokine receptor 2, Cancer, mutation, orthosteric and allosteric antagonists

2.

Cc Chemokine Receptor 2 is Allosterically Modulated by Sodium Ions and Amiloride Derivatives Through a Distinct Sodium Ion Binding Site

Number of pages: 29 Posted: 22 Mar 2024
Leiden University - Leiden Academic Centre for Drug Research, affiliation not provided to SSRN, Leiden University - Leiden Academic Centre for Drug Research, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Leiden University - Leiden Academic Centre for Drug Research, Leiden University - Leiden Academic Centre for Drug Research and Leiden University - Leiden Academic Centre for Drug Research
Downloads 57 (1,000,027)

Abstract:

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Chemokine receptor, sodium ion binding site, G protein-coupled receptor, allosterism