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Pierre-Luc Boudreault

Université de Sherbrooke

SCHOLARLY PAPERS

5

DOWNLOADS

208

TOTAL CITATIONS

0

Scholarly Papers (5)

1.

In Vitro and in Vivo Activity Profiles of Broad-Spectrum Bacterial Atp Synthase Inhibitors

Number of pages: 36 Posted: 29 Jun 2025
Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke and Université de Sherbrooke
Downloads 61 (951,658)

Abstract:

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Broad-spectrum antibiotics, Structure-activity relationship (SAR), Tomatidine analogs, ATP synthase inhibitors, Multidrug-resistant, Neutropenic mouse infection model, Drug Resistance

2.

From Garden to Lab: C-3 Chemical Modifications of Tomatidine Unveil Broad-Spectrum Atp Synthase Inhibitors to Combat Bacterial Resistance

Number of pages: 36 Posted: 21 Sep 2023
Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke and Université de Sherbrooke
Downloads 54 (1,031,043)

Abstract:

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Tomatidine, Antibacterial, Antibiotic resistance, ATP synthase inhibitors, Broad-spectrum

3.

Identification of ECM-Derived Skeletal Muscle Stem Cell Adhesion Motifs Using SPOT-Synthesis-Based Peptide Arrays

Number of pages: 51 Posted: 03 Nov 2023
Université de Sherbrooke, affiliation not provided to SSRN, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke, Université de Sherbrooke and Université de Sherbrooke
Downloads 40 (1,183,237)

Abstract:

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MuSCs, Satellite cells, myoblasts, Extracellular matrix, Stem cell niche, Adhesion motifs, Peptides

4.

Diversity-Oriented Synthesis of Second Generation Guanidinium-Rich Transporters Toward Cell-Selective Penetration

Number of pages: 27 Posted: 25 Oct 2024
affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN and Université de Sherbrooke
Downloads 29 (1,332,057)

Abstract:

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Guanidinium-Rich Transporters, Peptidomimetic, Solid-phase synthesis, Structure-activity relationships, Cell-penetrating peptides

5.

Structural Insights into Frog Skin-Derived Cyclic Peptides as Selective Matriptase Inhibitors

Number of pages: 35 Posted: 06 Sep 2025
affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Université de Sherbrooke, University of Gdansk, Université de Sherbrooke, Université de Sherbrooke and affiliation not provided to SSRN
Downloads 24 (1,399,036)

Abstract:

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Peptide inhibitors, proteases, matriptase, cyclic peptides, non-covalent inhibition, competitive inhibition, molecular dynamics simulations