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Maria Grazia Perrone

Università degli Studi di Bari “Aldo Moro” (UNIBA)

Italy

SCHOLARLY PAPERS

2

DOWNLOADS

88

TOTAL CITATIONS

0

Scholarly Papers (2)

1.

Synthesis and biological evaluation of novel fused pyridopyrimidine derivatives as topoisomerase I inhibitors and as potential antitumor agents: promising results in lung, ovary and gastric cancer

Number of pages: 55 Posted: 08 Jan 2026
affiliation not provided to SSRN, affiliation not provided to SSRN, Aarhus University, Aarhus University, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Università degli Studi di Bari “Aldo Moro” (UNIBA), Università degli Studi di Bari “Aldo Moro” (UNIBA), Università degli Studi di Bari “Aldo Moro” (UNIBA) and affiliation not provided to SSRN
Downloads 48 (1,097,529)

Abstract:

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pyrimidines, topoisomerase I, enzyme inhibition, antiproliferative effect

2.

Triazole-Benzodiazepine Derivatives: One-Pot Synthesis, Characterization, Hirshfeld Surface Analysis, Computational Insights and Anticancer Potential as Kif11 Inhibitors

Number of pages: 34 Posted: 27 Jul 2025
affiliation not provided to SSRN, Cadi Ayyad University, affiliation not provided to SSRN, Cadi Ayyad University, affiliation not provided to SSRN, Università degli Studi di Bari “Aldo Moro” (UNIBA), affiliation not provided to SSRN, affiliation not provided to SSRN, Università degli Studi di Bari “Aldo Moro” (UNIBA), Università degli Studi di Bari “Aldo Moro” (UNIBA) and Cadi Ayyad University
Downloads 40 (1,196,171)

Abstract:

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Cycloaddition Reaction, Characterization, DFT calculations, ADMET Studies, Anticancer Effects.