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Cinzia Tesauro

Aarhus University

Department of Biology

Section for Microbiology

Aarhus C, 8000

Denmark

SCHOLARLY PAPERS

2

DOWNLOADS

65

TOTAL CITATIONS

0

Scholarly Papers (2)

1.

Synthesis and biological evaluation of novel fused pyridopyrimidine derivatives as topoisomerase I inhibitors and as potential antitumor agents: promising results in lung, ovary and gastric cancer

Number of pages: 55 Posted: 08 Jan 2026
affiliation not provided to SSRN, affiliation not provided to SSRN, Aarhus University, Aarhus University, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Università degli Studi di Bari “Aldo Moro” (UNIBA), Università degli Studi di Bari “Aldo Moro” (UNIBA), Università degli Studi di Bari “Aldo Moro” (UNIBA) and affiliation not provided to SSRN
Downloads 48 (1,097,529)

Abstract:

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pyrimidines, topoisomerase I, enzyme inhibition, antiproliferative effect

2.

Exploring phosphorus substitution in chromeno[4,3-d]pyrido[1,2-a]pyrimidines: new insights into Topoisomerase 1 inhibition and cytotoxicity

Number of pages: 52 Posted: 08 Jul 2026
affiliation not provided to SSRN, Aarhus University, Aarhus University, affiliation not provided to SSRN and affiliation not provided to SSRN
Downloads 17

Abstract:

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pyrimidines, phosporous, topoisomerase 1, enzyme inhibition, antiproliferative effect