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Bernard Pirotte

University of Liège

Leige

Belgium

  • University of Liège

SCHOLARLY PAPERS

3

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87

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0

Scholarly Papers (3)

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1.

Exploring Thienothiadiazine Dioxides as Isosteric Analogues of Benzo- and Pyridothiadiazine Dioxides in the Search of New AMPA and Kainate Receptor Positive Allosteric Modulators

Number of pages: 42 Posted: 01 Nov 2023
Pierre Francotte, Yasmin Bay, Eric Goffin, Thomas Colson, Cindy Lesenfants, Jerzy Dorosz, Saara Laulumaa, Pierre Fraikin, Pascal de Tullio, Caroline Beaufour, Iuliana Botez, Darryl S. Pickering, Karla Frydenvang, Laurence Danober, Anders Skov Kristensen, Jette Sandholm Kastrup and Bernard Pirotte
University of Liège, University of Copenhagen, University of Liège, University of Liège, University of Liège, University of Copenhagen, University of Helsinki - Institute of Biotechnology, University of Liège, University of Liège, Institut de Recherches Servier, Institut de Recherches Servier, University of Copenhagen, University of Copenhagen, Institut de Recherches Servier, University of Copenhagen, University of Copenhagen and University of Liège
Downloads 35 (1,263,436)

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Ionotropic glutamate receptors, positive allosteric modulators, thieno[3, 2-e]-1, 2, 4-thiadiazine 1, 1-dioxides, 1, 2, 4-benzothiadiazine 1, 1-dioxides, X-ray crystallography, calcium-sensitive fluorescence-based assay

2.

Synthesis and Pharmacological Evaluation of Fluoro/Chloro-Substituted Acetyl and Benzoyl Esters of Quinine as Antimalarial Agents

Number of pages: 20 Posted: 30 Nov 2023
Jean-Gonfi Mvondo Mbala, Dani Thierry Mawete, Alain Nanikafuako Makiese, Prosper Lwanzo Kwiraviwe, Bibiche Kuyubuka Pangu, Eric Buini Nguimi, Richard Cimanga Kanyanga, Luc Pieters, Gilles Degotte, M. Frédérich, Aristote Matondo, Natascha Van Pelt, Guy Caljon, Bernard Pirotte, Blaise Mbala Mavinga and Sylvie-Mireille Bambi-Nyanguile
affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, University of Antwerp, University of Liège, University of Liège, Université de Kinshasa, University of Antwerp, University of Antwerp, University of Liège, affiliation not provided to SSRN and affiliation not provided to SSRN
Downloads 30 (1,332,057)

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quinine esters, antiplasmodial activity, Plasmodium falciparum

3.

Crystal Structure of the Gluk1 Ligand-Binding Domain with Kainate and the Full-Spanning Positive Allosteric Modulator Bpam538

Number of pages: 24 Posted: 24 Nov 2023
Yasmin Bay, Stine M. Frantsen, Darryl S. Pickering, Karla Frydenvang, Pierre Francotte, Bernard Pirotte, Anders Skov Kristensen and Jette Sandholm Kastrup
University of Copenhagen, affiliation not provided to SSRN, University of Copenhagen, University of Copenhagen, University of Liège, University of Liège, University of Copenhagen and University of Copenhagen
Downloads 22 (1,424,331)

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X-ray crystallography, ligand-binding domain of GluK1, positive allosteric modulator, kainate, binding mode