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Yu Jia

Fudan University

SCHOLARLY PAPERS

1

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44

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0

Scholarly Papers (1)

1.

Discovery of a High Potent PIM Kinase Inhibitor for Acute Myeloid Leukemia Based on N-Pyridinyl Amide Scaffold by Optimizing the Fragments Toward to Lys67 and Asp128/Glu171

Number of pages: 50 Posted: 24 Apr 2023
Fudan University, Fudan University, Fudan University, Fudan University - Department of Pharmaceutics, Fudan University, Fudan University, Fudan University - Department of Chemistry, SD Chem, Inc., ABA Chemicals Corporation, ABA Chemicals Corporation, Fudan University - Department of Chemistry and Fudan University - Department of Chemistry
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Abstract:

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N-pyridinyl amide scaffold, PIM inhibitors, Structure-activity relationship, Acute myeloid leukemia