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Jef Rozenski

KU Leuven

Oude Markt 13

Leuven, 3000

Belgium

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Scholarly Papers (1)

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Discovery and Exploration of Disubstituted [1,2,5]Oxadiazolo-[3,4-B]Pyrazines as Novel C-C Chemokine Receptor Type 5 Signaling Inhibitors Targeting the Intracellular Allosteric Binding Pocket

Number of pages: 57 Posted: 20 Dec 2024
Margaux Billen, Sten Reynders, Sandra Claes, Silke Kleinboelting, Jef Rozenski, Radu-George Bulai, Edoardo Rocca, Natalie Z M Homer, Scott P. Webster, Tim P. Kaminski, Eveline Lescrinier, Dominique Schols and Peter Verwilst
KU Leuven, KU Leuven, KU Leuven, affiliation not provided to SSRN, KU Leuven, KU Leuven, KU Leuven, Edinburgh Clinical Research Facility, affiliation not provided to SSRN, affiliation not provided to SSRN, KU Leuven, KU Leuven and KU Leuven
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Abstract:

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intracellular chemokine receptor antagonists, CCR5, SAR optimization, [1, 2, 5]oxadiazolo-[3, 4-b]pyrazines, binding mode validation