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Fengtao Zhou

Jinan University

Huang Pu Da Dao Xi 601, Tian He District

Guangzhou, 510632

China

SCHOLARLY PAPERS

3

DOWNLOADS

209

TOTAL CITATIONS

0

Scholarly Papers (3)

1.

Discovery of New Lenalidomide Derivatives as Potent and Selective Gspt1 Degraders

Number of pages: 35 Posted: 19 May 2023
Jinan University, Jinan University, Jinan University, Livzon Pharmaceutical Group Inc, Jinan University, Chinese Academy of Sciences (CAS), Jinan University, Jinan University and Jinan University
Downloads 113 (626,371)

Abstract:

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GSPT1, protein degradation, molecular glue, cancer

2.

Discovery of the First Potent Ror1 Degrader for the Treatment of Non-Small Cell Lung Cancer

Number of pages: 55 Posted: 13 Nov 2024
Jinan University, Jinan University, Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry, Jinan University, Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry, Jinan University, Chinese Academy of Sciences (CAS), Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CAS), Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry and Jinan University
Downloads 52 (1,041,696)

Abstract:

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ROR1, Pseudokinase, PROTACs, Protein Degradation, Apoptosis, Proliferation, NSCLC

3.

Discovery of 5-Aminopyrido[2,3- d]Pyrimidin-7(8 H)-One Derivatives as New Hematopoietic Progenitor Kinase 1 (HPK1) Inhibitors

Number of pages: 61 Posted: 30 Jan 2024
Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry, Jinan University, Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry, Jinan University, Chinese Academy of Sciences (CAS), Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CAS) and Chinese Academy of Sciences (CAS) - Shanghai Institute of Organic Chemistry
Downloads 44 (1,133,231)

Abstract:

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HPK1, Kinase inhibitor, Cancer immunotherapy, Selectivity, Cocrystal structure