default author photo

Samia M. Moustafa

Suez Canal University

SCHOLARLY PAPERS

2

DOWNLOADS

153

TOTAL CITATIONS

0

Scholarly Papers (2)

1.

Exploitation of Novel Pyrazolo[3,4-D]Pyrimidine Scaffold Tethered to Thiazole as Potential Egfr/Her2 Dual Kinase Inhibitor to Overcome Lapatinib Resistant Breast Cancer: Design, Synthesis, in Silico Docking and Molecular Dynamic Simulation

Number of pages: 62 Posted: 26 Feb 2025
Sphinx University, Zagazig University, Suez Canal University, Suez Canal University, King Abdulaziz University, King Abdulaziz University, King Abdulaziz University, King Abdulaziz University, Assiut University and King Abdulaziz University
Downloads 89 (753,595)

Abstract:

Loading...

Pyrazolo[3, 4-d]pyrimidine, Thiazoles, Lapatinib, EGFR, HER2, SKBr3, BT474, MDA-MB-453

2.

Development, Biological Evaluation, and Molecular Modelling of Novel Isocytosine and Guanidine Derivatives as Bace1 Inhibitors Using a Fragment Growing Strategy

Number of pages: 41 Posted: 13 Mar 2024
Badr university in Cairo, Zewail City of Science and Technology, Temple University, University of Sharjah, Suez Canal University, Suez Canal University, Zewail City of Science and Technology and Suez Canal University
Downloads 64 (924,743)

Abstract:

Loading...

Alzheimer's disease, BACE1 inhibitors, Aβ42, Molecular Modelling, Cranial/hepatic tissue safety