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Ismail Salama

Suez Canal University

SCHOLARLY PAPERS

2

DOWNLOADS

171

TOTAL CITATIONS

1

Scholarly Papers (2)

1.

Exploitation of Novel Pyrazolo[3,4-D]Pyrimidine Scaffold Tethered to Thiazole as Potential Egfr/Her2 Dual Kinase Inhibitor to Overcome Lapatinib Resistant Breast Cancer: Design, Synthesis, in Silico Docking and Molecular Dynamic Simulation

Number of pages: 62 Posted: 26 Feb 2025
Sphinx University, Zagazig University, Suez Canal University, Suez Canal University, King Abdulaziz University, King Abdulaziz University, King Abdulaziz University, King Abdulaziz University, Assiut University and King Abdulaziz University
Downloads 88 (753,595)

Abstract:

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Pyrazolo[3, 4-d]pyrimidine, Thiazoles, Lapatinib, EGFR, HER2, SKBr3, BT474, MDA-MB-453

2.

Development of 1, 2, 3-Triazole Hybrids as Multi-Faced Anticancer Agents Co-Targeting Egfr/Mtor Pathway and Tubulin Depolymerization

Number of pages: 51 Posted: 15 Nov 2024
Horus University, Suez Canal University, affiliation not provided to SSRN, affiliation not provided to SSRN and Suez Canal University
Downloads 83 (783,685)
Citation 1

Abstract:

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Colorectal cancer, 1, 2, 3-Triazole, Chalcones, Pyrazoles, Pyrimidines, EGFR/mTOR pathway, Tubulin Depolymerization, Cell Cycle Arrest, Commputational studies.