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Felice D. Kelly

Oregon Health and Science University

3181 S.W. Sam Jackson Park Rd.

Portland, OR 97201

United States

SCHOLARLY PAPERS

1

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87

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0

Scholarly Papers (1)

1.

DNA Pro-Retention Modulators of PARP1 Overcome Primary and Acquired Resistance to Clinical PARP Inhibitors

Number of pages: 48 Posted: 26 Sep 2025
Oregon Health and Science University, Oregon Health and Science University, University of Colorado at Boulder - Department of Biochemistry, University of Montreal, University of Pennsylvania, University of Pennsylvania, University of Pennsylvania, University of Montreal, University of Colorado at Boulder - Department of Biochemistry, University of Montreal, Oregon Health and Science University, Tilikum Therapeutics, Tilikum Therapeutics, Tilikum Therapeutics, Tilikum Therapeutics, Ludwig Maximilian University of Munich (LMU), Ludwig Maximilian University of Munich (LMU), University of Colorado at Boulder - Department of Biochemistry, University of Pennsylvania - Department of Biochemistry and Biophysics, University of Montreal, Oregon Health and Science University and Independent
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Abstract:

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Poly(ADP-ribose) polymerases (PARPs), NAD+-competitive inhibitors, Allosteric regulation, PARP inhibitor resistance, DNA damage response (DDR), Non-enzymatic functions, Synthetic lethality