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David Thal

Monash University - Drug Discovery Biology

Parkville, VIC 3052

Australia

SCHOLARLY PAPERS

2

DOWNLOADS

141

TOTAL CITATIONS

0

Scholarly Papers (2)

1.

Structural and Dynamic Mechanisms of Allostery at the M4 Muscarinic Acetylcholine Receptor

Number of pages: 79 Posted: 14 Feb 2022
Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Vanderbilt University - Department of Pharmacology, University of Glasgow - The Centre for Translational Pharmacology, Monash University - Drug Discovery Biology, University of Tokyo - Graduate School of Medicine, Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology and Monash University - Drug Discovery Biology
Downloads 111 (635,507)

Abstract:

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G protein coupled-receptor, M4 muscarinic acetylcholine receptor, allostery, cryoelectron microscopy, molecular dynamics, pharmacology, drug discovery

2.

Design, Synthesis and Evaluation of Novel 2-Phenyl-3-(1H-Pyrazol-4-yl)Pyridine Positive Allosteric Modulators for the M4 mAChR

Number of pages: 59 Posted: 04 May 2023
Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Drug Discovery Biology, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Monash Institute of Pharmaceutical Sciences, University of Glasgow - The Centre for Translational Pharmacology, Monash University - Drug Discovery Biology, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology and Monash University - Monash Institute of Pharmaceutical Sciences
Downloads 30 (1,318,317)

Abstract:

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acetylcholine, allosteric ligands, M4 muscarinic acetylcholine receptor, positive allosteric modulators, xanomeline