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Denise Wootten

Monash University - Drug Discovery Biology

Parkville, VIC 3052

Australia

SCHOLARLY PAPERS

3

DOWNLOADS

335

TOTAL CITATIONS

0

Scholarly Papers (3)

1.

Implications of Ligand-Receptor Binding Kinetics on GLP-1R Signalling

Number of pages: 26 Posted: 15 Jan 2022
Monash University - Drug Discovery Biology, affiliation not provided to SSRN, affiliation not provided to SSRN, Monash University - Drug Discovery Biology and Monash University - Drug Discovery Biology
Downloads 113 (630,858)

Abstract:

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Glucagon-like peptide-1 receptor, ligand binding kinetics, G protein activation kinetics, signalling kinetics, correlation

2.

Isoquinoline Small Molecule Ligands are Agonists and Probe-Dependent Allosteric Modulators of the Glucagon Subfamily of Gpcrs

Number of pages: 28 Posted: 22 May 2024
Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Monash Institute of Pharmaceutical Sciences, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology and Monash University - Drug Discovery Biology
Downloads 111 (635,507)

Abstract:

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GIPR, GLP1R, GCGR, CTR, class B1 GPCRs, allosteric modulation

3.

Structural and Dynamic Mechanisms of Allostery at the M4 Muscarinic Acetylcholine Receptor

Number of pages: 79 Posted: 14 Feb 2022
Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Vanderbilt University - Department of Pharmacology, University of Glasgow - The Centre for Translational Pharmacology, Monash University - Drug Discovery Biology, University of Tokyo - Graduate School of Medicine, Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology and Monash University - Drug Discovery Biology
Downloads 111 (635,507)

Abstract:

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G protein coupled-receptor, M4 muscarinic acetylcholine receptor, allostery, cryoelectron microscopy, molecular dynamics, pharmacology, drug discovery