Parkville, VIC 3052
Australia
Monash University - Drug Discovery Biology
G protein coupled-receptor, M4 muscarinic acetylcholine receptor, allostery, cryoelectron microscopy, molecular dynamics, pharmacology, drug discovery
G protein-coupled receptors (GPCRs)histamine H3 receptor (H3R)receptor isoformsbiased agonismligand biasneuromodulation
acetylcholine, allosteric ligands, M4 muscarinic acetylcholine receptor, positive allosteric modulators, xanomeline