default author photo

Celine Valant

Monash University - Drug Discovery Biology

Parkville, VIC 3052

Australia

SCHOLARLY PAPERS

3

DOWNLOADS

190

TOTAL CITATIONS

0

Scholarly Papers (3)

1.

Structural and Dynamic Mechanisms of Allostery at the M4 Muscarinic Acetylcholine Receptor

Number of pages: 79 Posted: 14 Feb 2022
Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology, Vanderbilt University - Department of Pharmacology, University of Glasgow - The Centre for Translational Pharmacology, Monash University - Drug Discovery Biology, University of Tokyo - Graduate School of Medicine, Monash University - Drug Discovery Biology, University of Kansas - Center for Computational Biology and Department of Molecular Biosciences, Monash University - Drug Discovery Biology and Monash University - Drug Discovery Biology
Downloads 111 (635,507)

Abstract:

Loading...

G protein coupled-receptor, M4 muscarinic acetylcholine receptor, allostery, cryoelectron microscopy, molecular dynamics, pharmacology, drug discovery

2.

Ligand-Directed Biased Agonism at Human Histamine H3 Receptor Isoforms Across Gαi/O- and Β-Arrestin2-Mediated Pathways

Number of pages: 74 Posted: 26 Oct 2023
Monash University - Monash Institute of Pharmaceutical Sciences, VU University Amsterdam, VU University Amsterdam, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology and Monash University - Monash Institute of Pharmaceutical Sciences
Downloads 49 (1,074,648)

Abstract:

Loading...

G protein-coupled receptors (GPCRs)histamine H3 receptor (H3R)receptor isoformsbiased agonismligand biasneuromodulation

3.

Design, Synthesis and Evaluation of Novel 2-Phenyl-3-(1H-Pyrazol-4-yl)Pyridine Positive Allosteric Modulators for the M4 mAChR

Number of pages: 59 Posted: 04 May 2023
Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Drug Discovery Biology, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Monash Institute of Pharmaceutical Sciences, University of Glasgow - The Centre for Translational Pharmacology, Monash University - Drug Discovery Biology, Monash University - Monash Institute of Pharmaceutical Sciences, Monash University - Drug Discovery Biology, Monash University - Drug Discovery Biology and Monash University - Monash Institute of Pharmaceutical Sciences
Downloads 30 (1,318,317)

Abstract:

Loading...

acetylcholine, allosteric ligands, M4 muscarinic acetylcholine receptor, positive allosteric modulators, xanomeline