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Aurélie Malzert-Fréon

Normandie Université

SCHOLARLY PAPERS

3

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129

TOTAL CITATIONS

0

Scholarly Papers (3)

New Antiplasmodial 4-Amino-Thieno[3,2-D]Pyrimidines with Improved Intestinal Permeability and Microsomal Stability

Number of pages: 30 Posted: 17 Sep 2022
University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), Aix Marseille Université, Sorbonne University, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille University, Sorbonne University, Sorbonne University, Normandie Université, Normandie Université, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université, UNIMES - Université de Nîmes - CHU de Nîmes (Centre Hospitalier Universitaire de Nîmes), Aix Marseille Université, Sorbonne University, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM) and University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM)
Downloads 33 (1,311,254)

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malaria, thienopyrimidine, erythocytic, hepatic, Plasmodium, solubility, permeability

New Antiplasmodial 4-Amino-Thieno[3,2-d]Pyrimidines with Improved Intestinal Permeability and Microsomal Stability

Number of pages: 30 Posted: 17 Sep 2022
University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), Aix Marseille Université, Sorbonne University, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille University, Sorbonne University, Sorbonne University, Normandie Université, Normandie Université, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université, UNIMES - Université de Nîmes - CHU de Nîmes (Centre Hospitalier Universitaire de Nîmes), Aix Marseille Université, Sorbonne University, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM) and University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM)
Downloads 25 (1,430,393)

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malaria, thienopyrimidine, erythocytic, hepatic, Plasmodium, solubility, permeability

2.

Synthesis of Antiplasmodial 2-Aminothieno[3,2-D]Pyrimidin-4(3h)-One Analogues Using the Scaffold Hopping Strategy

Number of pages: 30 Posted: 17 Jun 2022
Aix Marseille Université, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université, Sorbonne University, Sorbonne University, Sorbonne University, Normandie Université, Normandie Université, Normandie Université, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), UNIMES - Université de Nîmes - CHU de Nîmes (Centre Hospitalier Universitaire de Nîmes), Sorbonne University, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université and Aix Marseille Université
Downloads 40 (1,182,860)

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Malaria, Plasmodium, scaffold hopping, thienopyrimidinone

3.

Novel Thienopyrimidones Targeting Hepatic and Erythrocytic Stages of Plasmodium Parasites with Increased Microsomal Stability

Number of pages: 33 Posted: 20 Jul 2023
University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), Aix Marseille Université, Sorbonne University, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille University, Sorbonne University, Sorbonne University, Normandie Université, Normandie Université, Normandie Université, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université, University Grenoble Alpes, Aix Marseille Université, Sorbonne University, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM) and University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM)
Downloads 31 (1,304,153)

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Malaria, Thienopyrimidine, Erythocytic, Hepatic, Plasmodium, Microsomal Stability, Permeability