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Sophie Corvaisier

Normandie Université

SCHOLARLY PAPERS

5

DOWNLOADS

236

TOTAL CITATIONS

0

Scholarly Papers (5)

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1.

ID Card of Mcl-1 PROTAC degrader: From in silico design to biological validation in chemoresistant ovarian cancer

Number of pages: 66 Posted: 01 Dec 2025
Marie Cornu, Jocelyn Pezeril, Nicolas Guedeney, Hippolyte Paysant, Thomas Lemaitre, Florian Schwalen, Romane Florent, Julie N’Guyen, Sophie Corvaisier, Marc Since, Dimitri Fayolle, Amina Hamza, Mike Maillasson, Jana Sopkova de Oliveira Santos, Charline Kieffer, Laurent Poulain and anne sophie voisin-chiret
affiliation not provided to SSRN, affiliation not provided to SSRN, Université Paris Cité, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Normandie Université, Normandie Université, Université de Lyon, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN and University of Caen Normandy
Downloads 62 (942,311)

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PROTAC, Targeted protein degradation, Mcl-1, ovarian cancer, oligopyridine

2.

New Antiplasmodial 4-Amino-Thieno[3,2-D]Pyrimidines with Improved Intestinal Permeability and Microsomal Stability

Downloads 58 (979,888)

New Antiplasmodial 4-Amino-Thieno[3,2-D]Pyrimidines with Improved Intestinal Permeability and Microsomal Stability

Number of pages: 30 Posted: 17 Sep 2022
Prisca Lagardère, Romain Mustière, Nadia Amanzougaghene, Sébastien Hutter, Marion Casanova, Jean-François Franetich, Shahin Tajeri, Aurélie Malzert-Fréon, Sophie Corvaisier, Nadine Azas, Patrice Vanelle, Pierre Verhaeghe, Nicolas Primas, Dominique Mazier, Nicolas Masurier and Vincent Lisowski
University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), Aix Marseille Université, Sorbonne University, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille University, Sorbonne University, Sorbonne University, Normandie Université, Normandie Université, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université, UNIMES - Université de Nîmes - CHU de Nîmes (Centre Hospitalier Universitaire de Nîmes), Aix Marseille Université, Sorbonne University, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM) and University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM)
Downloads 33 (1,311,254)

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malaria, thienopyrimidine, erythocytic, hepatic, Plasmodium, solubility, permeability

New Antiplasmodial 4-Amino-Thieno[3,2-d]Pyrimidines with Improved Intestinal Permeability and Microsomal Stability

Number of pages: 30 Posted: 17 Sep 2022
Prisca Lagardère, Romain Mustière, Nadia Amanzougaghene, Sébastien Hutter, Marion Casanova, Jean-François Franetich, Shahin Tajeri, Aurélie Malzert-Fréon, Sophie Corvaisier, Nadine Azas, Patrice Vanelle, Pierre Verhaeghe, Nicolas Primas, Dominique Mazier, Nicolas Masurier and Vincent Lisowski
University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), Aix Marseille Université, Sorbonne University, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille University, Sorbonne University, Sorbonne University, Normandie Université, Normandie Université, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université, UNIMES - Université de Nîmes - CHU de Nîmes (Centre Hospitalier Universitaire de Nîmes), Aix Marseille Université, Sorbonne University, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM) and University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM)
Downloads 25 (1,430,393)

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malaria, thienopyrimidine, erythocytic, hepatic, Plasmodium, solubility, permeability

3.

Synthesis, in Vitro and in Vivo Biological Evaluation of Novel Dual Compounds Targeting Both Acetylcholinesterase and Serotonergic 5-Ht4 Receptors with Potential Interest in Alzheimer's Disease Treatment

Number of pages: 77 Posted: 03 Oct 2024
Patrick Dallemagne, Christophe Rochais, Cédric Lecoutey, Julien Lalut, Audrey Davis, Emilie Duval, Florence Gaven, Stacy Largillière, Gérald Née, Sophie Corvaisier, Jana Sopkova de Oliveira Santos, Marc Since, Thomas Freret, Romain Legrand, Noëlle Callizot, Sylvie Claeysen and Michel Boulouard
affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Normandie Université, affiliation not provided to SSRN, Normandie Université, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN and affiliation not provided to SSRN
Downloads 45 (1,120,871)

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Alzheimer's disease, Pleiotropic, acetylcholinesterase, Serotonin, 5-HT4

4.

Synthesis of Antiplasmodial 2-Aminothieno[3,2-D]Pyrimidin-4(3h)-One Analogues Using the Scaffold Hopping Strategy

Number of pages: 30 Posted: 17 Jun 2022
Romain Mustière, Prisca Lagardère, Sébastien Hutter, Viviana Dell'Orco, Nadia Amanzougaghene, Shahin Tajeri, Jean-François Franetich, Sophie Corvaisier, Marc Since, Aurélie Malzert-Fréon, Nicolas Masurier, Vincent Lisowski, Pierre Verhaeghe, Dominique Mazier, Nadine Azas, Patrice Vanelle and Nicolas Primas
Aix Marseille Université, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université, Sorbonne University, Sorbonne University, Sorbonne University, Normandie Université, Normandie Université, Normandie Université, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), UNIMES - Université de Nîmes - CHU de Nîmes (Centre Hospitalier Universitaire de Nîmes), Sorbonne University, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université and Aix Marseille Université
Downloads 40 (1,182,860)

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Malaria, Plasmodium, scaffold hopping, thienopyrimidinone

5.

Novel Thienopyrimidones Targeting Hepatic and Erythrocytic Stages of Plasmodium Parasites with Increased Microsomal Stability

Number of pages: 33 Posted: 20 Jul 2023
Prisca Lagardère, Romain Mustière, Nadia Amanzougaghene, Sébastien Hutter, Marion Casanova, Jean-François Franetich, Shahin Tajeri, Aurélie Malzert-Fréon, Sophie Corvaisier, Marc Since, Nadine Azas, Patrice Vanelle, Pierre Verhaeghe, Nicolas Primas, Dominique Mazier, Nicolas Masurier and Vincent Lisowski
University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM), Aix Marseille Université, Sorbonne University, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille University, Sorbonne University, Sorbonne University, Normandie Université, Normandie Université, Normandie Université, Aix Marseille University - UMR VITROME - Tropical Eukaryotic Pathogens, Aix Marseille Université, University Grenoble Alpes, Aix Marseille Université, Sorbonne University, University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM) and University of Montpellier - Institut des Biomolécules Max Mousseron (IBMM)
Downloads 31 (1,304,153)

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Malaria, Thienopyrimidine, Erythocytic, Hepatic, Plasmodium, Microsomal Stability, Permeability