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Rafael Dolezal

University Hospital Hradec Kralove

SCHOLARLY PAPERS

3

DOWNLOADS

132

TOTAL CITATIONS

0

Scholarly Papers (3)

1.

Highly Selective Butyrylcholinesterase Inhibitors Related to Amaryllidaceae Alkaloids - Design, Synthesis, and Biological Evaluation

Number of pages: 62 Posted: 03 Mar 2023
Charles University, Charles University, Charles University, Charles University, Place Général Valérie André, Place Général Valérie André, Place Général Valérie André, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Defence, Trebesska - Faculty of Military Health Sciences, Charles University, Charles University, Charles University, University Hospital Hradec Kralove and Charles University
Downloads 60 (961,006)

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Alzheimer's disease, Amaryllidaceae alkaloids, butyrylcholinesterase, cholinesterase inhibitors, crystallographic study, qsar

2.

Rational Design, Synthesis and Evaluation of Piperazine Derivatives as Promising Radioprotective Agents: Toward Next-Generation Alternatives to Amifostine

Number of pages: 35 Posted: 28 Jul 2025
affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove and University Hospital Hradec Kralove
Downloads 36 (1,236,159)

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Radioprotection, Drug design, radiation, radiation medical countermeasures, piperazine, in vitro

3.

2,6-Disubstituted 7-(Naphthalen-2-Ylmethyl)-7h-Purines as a New Class of Potent Antitubercular Agents Inhibiting Dpre1

Number of pages: 85 Posted: 18 May 2023
University Hospital Hradec Kralove, University of Defence in Brno, Comenius University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, Charles University, University Hospital Hradec Kralove, Eötvös Loránd University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Chemistry and Technology, Prague, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, Charles University, Charles University, Eötvös Loránd University, Comenius University, University of Lille - CHU Lille, Charles University and University Hospital Hradec Kralove
Downloads 36 (1,249,711)

Abstract:

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Tuberculosis, purine, Mycobacterium tuberculosis, DprE1, Structure-activity relationships