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Lubica Muckova

University Hospital Hradec Kralove

SCHOLARLY PAPERS

5

DOWNLOADS

233

TOTAL CITATIONS

0

Scholarly Papers (5)

1.

Privileged Multi-Target Directed Propargyl-Tacrines Combining Cholinesterase and Monoamine Oxidase Inhibition Activities

Number of pages: 37 Posted: 14 Mar 2022
affiliation not provided to SSRN, affiliation not provided to SSRN, University of Hradec Králové, affiliation not provided to SSRN, affiliation not provided to SSRN, University Hospital Hradec Kralove, affiliation not provided to SSRN, University Hospital Hradec Kralove, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN and affiliation not provided to SSRN
Downloads 67 (899,324)

Abstract:

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Cholinesterase inhibitor, Alzheimer's disease, Monoamine oxidase inhibitor, Propargyl amines, Tacrine

2.

Novel Antitubercular Agents Based on 2,4-Disubstituted 5-(Aryl-2-Ylmethyl)-5h-Pyrrolo[3,2-D]Pyrimidines

Number of pages: 74 Posted: 19 Jun 2025
affiliation not provided to SSRN, University of Pardubice, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, affiliation not provided to SSRN, University Hospital Hradec Kralove, University of Pardubice, University of Pardubice, University Hospital Hradec Kralove, affiliation not provided to SSRN, affiliation not provided to SSRN, Academy of Sciences of the Czech Republic, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Medical University of Gdansk, Medical University of Gdansk, University Hospital Hradec Kralove, Charles University, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN and University Hospital Hradec Kralove
Downloads 57 (989,921)

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deazapurine, Mycobacterium tuberculosis, pyrrole, pyrimidine, tuberculosis

3.

Carltonine-Derived Compounds for Targeted Butyrylcholinesterase Inhibition

Number of pages: 43 Posted: 28 Nov 2023
Charles University, Charles University, Charles University, Charles University, University Hospital Hradec Kralove, Charles University, Charles University, affiliation not provided to SSRN, University of Defence in Brno, University of Defense, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Defence, Trebesska - Faculty of Military Health Sciences, University Hospital Hradec Kralove and Charles University
Downloads 46 (1,109,210)

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Alzheimer's disease, Amaryllidaceae alkaloids, acetylcholinesterase, butyrylcholinesterase, cholinesterase inhibitors

4.

2,6-Disubstituted 7-(Naphthalen-2-Ylmethyl)-7h-Purines as a New Class of Potent Antitubercular Agents Inhibiting Dpre1

Number of pages: 85 Posted: 18 May 2023
University Hospital Hradec Kralove, University of Defence in Brno, Comenius University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, Charles University, University Hospital Hradec Kralove, Eötvös Loránd University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Chemistry and Technology, Prague, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, Charles University, Charles University, Eötvös Loránd University, Comenius University, University of Lille - CHU Lille, Charles University and University Hospital Hradec Kralove
Downloads 37 (1,249,711)

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Tuberculosis, purine, Mycobacterium tuberculosis, DprE1, Structure-activity relationships

5.

Carltonine B Derivatives: Synthesis and Structure-Activity Relationship Insights for Selective Butyrylcholinesterase Inhibition

Number of pages: 53 Posted: 19 Feb 2026
affiliation not provided to SSRN, affiliation not provided to SSRN, University Hospital Hradec Kralove, University of Defense, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Defence, Trebesska - Faculty of Military Health Sciences, University Hospital Hradec Kralove, Jagiellonian University in Krakow - Faculty of Pharmacy, affiliation not provided to SSRN, University Hospital Hradec Kralove, University of Caen Normandy, affiliation not provided to SSRN, affiliation not provided to SSRN, Charles University and University Hospital Hradec Kralove
Downloads 26 (1,411,822)

Abstract:

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Amaryllidaceae alkaloid, Alzheimer's Disease, butyrylcholinesterase, Enzyme inhibition, cytotoxicity