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Katarína Mikušová

Comenius University

Slovakia

SCHOLARLY PAPERS

2

DOWNLOADS

75

TOTAL CITATIONS

0

Scholarly Papers (2)

1.

Side Chain-Modified Benzothiazinone Derivatives with Anti-Mycobacterial Activity

Number of pages: 31 Posted: 01 Dec 2022
Soochow University, Capital Medical University - Beijing Chest Hospital, University of Pavia, Comenius University, Russian Academy of Sciences (RAS) - Research Center of Biotechnology, Soochow University, Soochow University, Comenius University, Russian Academy of Sciences (RAS) - Research Center of Biotechnology, University of Pavia, Capital Medical University - Beijing Chest Hospital, Soochow University and Soochow University - College of Pharmaceutical Sciences
Downloads 38 (1,222,651)

Abstract:

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Anti-tubercular agents, DprE1 inhibitor, Benzothiazinone analogs, Structure activity relationship, in vivo activity

2.

2,6-Disubstituted 7-(Naphthalen-2-Ylmethyl)-7h-Purines as a New Class of Potent Antitubercular Agents Inhibiting Dpre1

Number of pages: 85 Posted: 18 May 2023
University Hospital Hradec Kralove, University of Defence in Brno, Comenius University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, Charles University, University Hospital Hradec Kralove, Eötvös Loránd University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Chemistry and Technology, Prague, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, Charles University, Charles University, Eötvös Loránd University, Comenius University, University of Lille - CHU Lille, Charles University and University Hospital Hradec Kralove
Downloads 37 (1,249,711)

Abstract:

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Tuberculosis, purine, Mycobacterium tuberculosis, DprE1, Structure-activity relationships