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Martin Novák

Charles University

SCHOLARLY PAPERS

3

DOWNLOADS

146

TOTAL CITATIONS

0

Scholarly Papers (3)

1.

Novel Antitubercular Agents Based on 2,4-Disubstituted 5-(Aryl-2-Ylmethyl)-5h-Pyrrolo[3,2-D]Pyrimidines

Number of pages: 74 Posted: 19 Jun 2025
affiliation not provided to SSRN, University of Pardubice, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, affiliation not provided to SSRN, University Hospital Hradec Kralove, University of Pardubice, University of Pardubice, University Hospital Hradec Kralove, affiliation not provided to SSRN, affiliation not provided to SSRN, Academy of Sciences of the Czech Republic, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Medical University of Gdansk, Medical University of Gdansk, University Hospital Hradec Kralove, Charles University, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN and University Hospital Hradec Kralove
Downloads 57 (989,921)

Abstract:

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deazapurine, Mycobacterium tuberculosis, pyrrole, pyrimidine, tuberculosis

2.

Phenoxytacrine Derivatives: Low-Toxicity Neuroprotectants Exerting Affinity to Ifenprodil-Binding Site and Cholinesterase Inhibition

Number of pages: 49 Posted: 19 Dec 2023
Czech Academy of Sciences, University Hospital Hradec Kralove, Institute of Experimental Medicine of the CAS, National Institute of Mental Health, Czech Republic, National Institute of Mental Health, Czech Republic, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, University of Defence in Brno, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, National Institute of Mental Health, Czech Republic, Institute of Experimental Medicine of the CAS, Institute of Experimental Medicine of the CAS, Institute of Experimental Medicine of the CAS, University Hospital Hradec Kralove, University of Oslo, Government of the United States of America - National Institute of Mental Health, Czech Academy of Sciences and University Hospital Hradec Kralove
Downloads 53 (1,031,043)

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Alzheimer´s disease; electrophysiology; glutamate receptor; acetylcholinesterase; neuroprotection; in vivo; Tacrine

3.

2,6-Disubstituted 7-(Naphthalen-2-Ylmethyl)-7h-Purines as a New Class of Potent Antitubercular Agents Inhibiting Dpre1

Number of pages: 85 Posted: 18 May 2023
University Hospital Hradec Kralove, University of Defence in Brno, Comenius University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, Charles University, University Hospital Hradec Kralove, Eötvös Loránd University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Chemistry and Technology, Prague, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, Charles University, Charles University, Eötvös Loránd University, Comenius University, University of Lille - CHU Lille, Charles University and University Hospital Hradec Kralove
Downloads 36 (1,249,711)

Abstract:

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Tuberculosis, purine, Mycobacterium tuberculosis, DprE1, Structure-activity relationships