default author photo

Martin Kufa

University Hospital Hradec Kralove

SCHOLARLY PAPERS

3

DOWNLOADS

153

TOTAL CITATIONS

0

Scholarly Papers (3)

1.

Highly Selective Butyrylcholinesterase Inhibitors Related to Amaryllidaceae Alkaloids - Design, Synthesis, and Biological Evaluation

Number of pages: 62 Posted: 03 Mar 2023
Charles University, Charles University, Charles University, Charles University, Place Général Valérie André, Place Général Valérie André, Place Général Valérie André, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Defence, Trebesska - Faculty of Military Health Sciences, Charles University, Charles University, Charles University, University Hospital Hradec Kralove and Charles University
Downloads 60 (961,006)

Abstract:

Loading...

Alzheimer's disease, Amaryllidaceae alkaloids, butyrylcholinesterase, cholinesterase inhibitors, crystallographic study, qsar

2.

Novel Antitubercular Agents Based on 2,4-Disubstituted 5-(Aryl-2-Ylmethyl)-5h-Pyrrolo[3,2-D]Pyrimidines

Number of pages: 74 Posted: 19 Jun 2025
affiliation not provided to SSRN, University of Pardubice, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, affiliation not provided to SSRN, University Hospital Hradec Kralove, University of Pardubice, University of Pardubice, University Hospital Hradec Kralove, affiliation not provided to SSRN, affiliation not provided to SSRN, Academy of Sciences of the Czech Republic, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, Medical University of Gdansk, Medical University of Gdansk, University Hospital Hradec Kralove, Charles University, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN, affiliation not provided to SSRN and University Hospital Hradec Kralove
Downloads 57 (989,921)

Abstract:

Loading...

deazapurine, Mycobacterium tuberculosis, pyrrole, pyrimidine, tuberculosis

3.

2,6-Disubstituted 7-(Naphthalen-2-Ylmethyl)-7h-Purines as a New Class of Potent Antitubercular Agents Inhibiting Dpre1

Number of pages: 85 Posted: 18 May 2023
University Hospital Hradec Kralove, University of Defence in Brno, Comenius University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, Charles University, University Hospital Hradec Kralove, Eötvös Loránd University, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University of Chemistry and Technology, Prague, University Hospital Hradec Kralove, University Hospital Hradec Kralove, University Hospital Hradec Kralove, Charles University, University Hospital Hradec Kralove, Charles University, Charles University, Eötvös Loránd University, Comenius University, University of Lille - CHU Lille, Charles University and University Hospital Hradec Kralove
Downloads 36 (1,249,711)

Abstract:

Loading...

Tuberculosis, purine, Mycobacterium tuberculosis, DprE1, Structure-activity relationships